7-Hydroxyflavone 7羟基黄酮
产品介绍
7-Hydroxyflavone是从臭茉莉中分离的一种口服活性黄酮类化合物,具有显著的抗炎活性。它通过激活ERK/Nrf2/HO-1信号通路保护肾细胞免受尼古丁损伤,并能有效抑制PKM2(IC50=2.12 μM)、COX-2(IC50=27µg/mL)和5-LOX(IC50=33µg/mL)等关键靶点。
产品性质
产品特色
/
存储条件
-25~-15℃避光保存,有效期3年。
COA
已发表文献
[1] Sengupta B, Sahihi M, Dehkhodaei M, Kelly D, Arany I. Differential roles of 3-Hydroxyflavone and 7-Hydroxyflavone against nicotine-induced oxidative stress in rat renal proximal tubule cells. PLoS One. 2017 Jun 22;12(6):e0179777. doi: 10.1371/journal.pone.0179777. PMID: 28640852; PMCID: PMC5480997.[2]LI W, WANG X, SUN Y, et al. 7-Hydroxyflavone confers cardioprotection against myocardial ischemia/reperfusion injury in rats via inhibition of MAPK/NF-κB pathway[J]. International Journal of Molecular Medicine, 2018, 42(4): 2053-2064.
相关产品
推荐应用
联系我们





