Kuwanon G是一种黄酮类化合物,可作为蛙皮素受体拮抗剂。Kuwanon G具有抗菌、抗肿瘤、抗炎、抗氧化、抗动脉粥样硬化及神经保护等多种生物活性。Kuwanon G桑黄酮G对口腔致病菌(尤其是致龋菌和牙周病原菌)表现出较强的抑制能力,并能诱导肿瘤细胞凋亡,抑制其增殖、迁移和侵袭。Kuwanon G适用于胃癌及动脉粥样硬化等相关疾病的研究。
[1] Geng Z,Yang J,Niu M,Liu X,Shi J,Liu Y,Yao X,Zhang Y,Zhang X,Hu J.[Kuwanon G inhibits growth,migration and invasion of gastric cancer cells by regulating the PI3K/AKT/mTOR pathway].Nan Fang Yi Ke Da Xue Xue Bao.2024 Aug 20;44(8):1476-1484.Chinese.doi:10.12122/j.issn.1673-4254.2024.08.06.PMID:39276043;PMCID:PMC11378037.[2]Liu XX,Zhang XW,Wang K,Wang XY,Ma WL,Cao W,Mo D,Sun Y,Li XQ.Kuwanon G attenuates atherosclerosis by upregulation of LXRα-ABCA1/ABCG1 and inhibition of NFκB activity in macrophages.Toxicol Appl Pharmacol.2018 Feb 15;341:56-63.doi:10.1016/j.taap.2018.01.007.Epub 2018 Feb 2.PMID:29355567.





